发明名称 |
NOVEL SULFONYL DERIVATIVES |
摘要 |
Sulfonyl derivatives represented by the following general formula (I): Q1-Q2 - T1-Q3-SO2-QA and drugs containing the same (wherein Q1 is an optionally substituted, saturated or unsaturated, five- or six-membered cyclic hydrocarbon group, a five- or six-membered heterocyclic group, or the like; Q2 is a single bond, oxygen, sulfur, C1-C6 alkylene or the like; QA is optional ly substituted arylalkenyl, heteroarylalkenyl or the like; and T1 is carbonyl o r the like). These compounds have potent FXa-inhibitory effects and promptly exert satisfactory and persistent antithrombotic effects through oral administration, thus being useful as anticoagulant agents little accompanied with side effects.
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申请公布号 |
CA2340100(A1) |
申请公布日期 |
2000.02.24 |
申请号 |
CA19992340100 |
申请日期 |
1999.08.11 |
申请人 |
DAIICHI PHARMACEUTICAL CO., LTD. |
发明人 |
KOBAYASHI, SYOZO;HAGINOYA, NORIYASU;SUZUKI, MASANORI;KOMORIYA, SATOSHI;NAGATA, TSUTOMU;ITO, MASAYUKI;NAGAHARA, TAKAYASU;MOCHIZUKI, AKIYOSHI;HORINO, HARUHIKO;YOSHINO, TOSHIHARU |
分类号 |
A61P7/02;C07D207/08;C07D207/12;C07D207/22;C07D211/34;C07D211/70;C07D213/56;C07D213/61;C07D213/73;C07D213/75;C07D213/82;C07D213/84;C07D213/89;C07D233/18;C07D233/54;C07D233/64;C07D233/88;C07D239/42;C07D239/48;C07D243/08;C07D277/28;C07D277/40;C07D401/04;C07D401/10;C07D401/12;C07D401/14;C07D405/04;C07D405/12;C07D409/04;C07D409/12;C07D409/14;C07D417/04;C07D417/12;C07D417/14;C07D491/048;(IPC1-7):C07D207/04;C07D471/04;C07D495/04;C07D498/04;C07D513/04;C07D235/08;C07D295/22;C07D217/26;C07D233/26;A61K31/415;A61K31/435;C07D209/44;A61K31/44;A61K31/445;A61K31/47;C07D215/48;A61K31/495;A61K31/505;A61K31/53;A61K31/535;A61K31/54;A61K31/55;C07D333/68;C07D307/85 |
主分类号 |
A61P7/02 |
代理机构 |
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