发明名称 AZETIDINE DERIVATIVES USEFUL IN TREATING PAIN, DIABETES AND DISORDERS OF LIPID METABOLISM
摘要 Disclosed are compounds of the formula: and compounds of the formula: wherein R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>5</SUP>, u and v are as defined herein. Also disclosed are methods of treating pain (e.g., inflammatory pain, chronic pain, and neuropathic pain), methods of treating diabetes, and methods of inhibiting the absorption of cholesterol using compounds of formula I or IIA.
申请公布号 US2008089858(A1) 申请公布日期 2008.04.17
申请号 US20070854600 申请日期 2007.09.13
申请人 MCKITTRICK BRIAN A;SMITH ELIZABETH M;BENNETT CHAD E;HARRIS JOEL M;KISELGOF EUGENIA Y;KNUTSON CHAD E;KORAKAS PETER;TULSHIAN DEEN;KIM HYUNJIN 发明人 MCKITTRICK BRIAN A.;SMITH ELIZABETH M.;BENNETT CHAD E.;HARRIS JOEL M.;KISELGOF EUGENIA Y.;KNUTSON CHAD E.;KORAKAS PETER;TULSHIAN DEEN;KIM HYUNJIN
分类号 A61K31/438;A61K31/565;A61K31/57;A61K31/573;A61K31/675;A61K38/20;A61P3/10;C07D471/10 主分类号 A61K31/438
代理机构 代理人
主权项
地址