发明名称 HIV PROTEASE INHIBITORS FOR TREATING OF HIV INFECTIONS AND A PHARMACEUTICAL COMPOSITION THEREOF
摘要 Phosphonate substituted compounds with HIV protease inhibitory properties having use as therapeutics and for other industrial purposes are disclosed according to a general structure formulaThe compositions, comprising compounds according to the invention, inhibit 5 HIV protease activity and/or are useful therapeutically for the treatment of AIDS and other antiviral infections, as well as in assays for the detection of HIV protease.
申请公布号 EA008775(B1) 申请公布日期 2007.08.31
申请号 EA20040001436 申请日期 2003.04.25
申请人 GILEAD SCIENCE, INC. 发明人 BECKER MARK, M.;BRYANT CLIFFORD;WANG JIANYING;DASTGAN AZAR;JIN HAOLUN;KIM CHOUNG, U.;LEE CHRISTOPHER, P.;LEE WILLIAM, A.;LIN KUEI-YING;LIU HONGTAO;MITCHELL MICHAEL, L.;MACKMAN RICHARD, L.;NELSON PETER, H.;PYUN HYUNG-JUNG;ROWE TANISHA, D.;SWAMINATHAN SUNDARAMOORTHI;SPARACINO MARK;XU LIANHONG;TARIO JAMES, D.;WILLIAMS MATTHEW, A.;FARDIS MARIA;HE GONG-XIN;CHEN JAMES, M.;CHEN XIAOWU;ZHANG LIJUN;ZHANG JIANCUN;ARIMILLI MURTY, N.;YU RICHARD, H.;YANG ZHENG-YU
分类号 C07F9/40;C12N9/99;A61K31/4155;A61K31/66;A61K31/665;A61K31/675;A61P31/18;A61P43/00;C07D213/75;C07D213/85;C07D231/12;C07D231/20;C07D233/42;C07D239/48;C07D239/80;C07D243/04;C07D265/18;C07D307/68;C07D401/06;C07D403/06;C07D471/14;C07D491/04;C07F;C07F9/02;C07F9/38;C07F9/44;C07F9/58;C07F9/62;C07F9/645;C07F9/6506;C07F9/6509;C07F9/6512;C07F9/653;C07F9/6533;C07F9/655;C07F9/6558;C07F9/6561;C07F9/6584;C12N9/16;C12Q1/18;C12Q1/37;C12Q1/44;C12Q1/70;G01N33/04;G01N33/50 主分类号 C07F9/40
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