Azole derivative, method for producing same, intermediate compound, and agricultural or horticultural chemical agent and industrial material protecting agent

摘要

Provided is an azole derivative superior in disease-controlling activity contained as an active ingredient in agricultural or horticultural chemical agents.;The azole derivative according to the present invention is represented by the following General Formula (I):;
(in Formula (I), R1 represents an unsubstituted or substituted C1-C6-alkyl group;

R2 represents a carbonyl group-containing functional group, wherein the carbon atom in the carbonyl group is bound to the carbon atom in the cyclopentane ring substituted with R1 and to a hydrogen atom, a hydroxyl group, R3, OR3, or NR3R4;

R3 and R4 each represent a C1-C6-alkyl group, a C2-C6-alkenyl group, or a C2-C6-alkynyl group;

Y represents a halogen atom, a C1-C4-alkyl group, a C1-C4-haloalkyl group, a C1-C4-alkoxy group, a C1-C4-haloalkoxy group, a phenyl group, a cyano group, or a nitro group;

m is 0 to 5; and

A represents a nitrogen atom or a methine group).

主权项

1. An intermediate compound of Formula (XI) wherein Y represents a halogen atom, a C1-C4-alkyl group, a C1-C4-haloalkyl group, a C1-C4-alkoxy group, a C1-C4-haloalkoxy group, a phenyl group, a cyano group, or a nitro group; m is 0 to 5; n is 1 to 6; and A represents a nitrogen atom or a methine group; R3 represents a hydrogen atom, a C1-C6-alkyl group, a C2-C6-alkenyl group, or a C2-C6-alkynyl group wherein the intermediate compound is used for the production of an azole derivative represented by the following General Formula (I):wherein R1 represents a halogen atom-substituted C1-C6-alkyl group;
R2 represents COOR3, wherein the carbon atom in the carbonyl group is bound to the carbon atom in the cyclopentane ring substituted with R1; R3 and R4 each represent a hydrogen atom, a C1-C6-alkyl group, a C2-C6-alkenyl group, or a C2-C6-alkynyl group; and Y, m, and A are as defined above.