发明名称 |
METHOD FOR THE PRODUCTION OF TELMISARTAN |
摘要 |
The invention relates to a novel method for the production of telmisartan by reacting 2-n-propyl-4-methyl-6- (1'-methylbenzimidazol-2'-yl)-benzimidazol with a compound of general formula (IV), in which Z is a leaving group, wherein the compound 2-cyano-4'-[2''-n-propyl-4''-methyl-6'' -(1'''-methylbenzimidazol-2'''-yl) benzimidazol-1''-ylmethyl]biphenyl is obtained, and subsequently conducting hydrolysis of the nitrile to acid function.
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申请公布号 |
KR20050118699(A) |
申请公布日期 |
2005.12.19 |
申请号 |
KR20057018333 |
申请日期 |
2004.03.26 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
HAUEL NORBERT;DACH ROLF;HEITGER HELMUT;MEYER OLIVER |
分类号 |
C07D235/04;C07D235/18;C07D403/02;C07D403/04;(IPC1-7):C07D403/04 |
主分类号 |
C07D235/04 |
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