发明名称 |
NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES. |
摘要 |
DISCLOSED ARE NOVEL CATHEPSIN S, K, F, L AND B REVERSIBLE INHIBITORY COMPOUNDS OF THE FORMULAS (1), (11), (1A) AND (1B) FURTHER DEFINED HEREIN. THE COMPOUNDS ARE USEFUL FOR TREATING AUTOIMMUNE DISEASES. ALSO DISCLOSED ARE PROCESSES FOR MAKING SUCH NOVEL COMPOUNDS.
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申请公布号 |
MY122696(A) |
申请公布日期 |
2006.04.29 |
申请号 |
MYPI20004216 |
申请日期 |
2000.09.11 |
申请人 |
BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. |
发明人 |
MICHEL JOSE EMMANUEL;ERICK RICHARD ROUSH YOUNG;LEAH LYNN FRYE;EUGENE RICHARD HICKEY;WEIMIN LIU;TINA MARIE MORWICK;DENICE MARY SPERO;SANXING SUN;DAVID S. THOMSON;YANCEY DAVID WARD |
分类号 |
A61K31/535;A61K31/428;A61K31/4468;A61K31/4535;A61K31/454;A61K31/495;A61K31/496;A61K31/4965;A61K31/506;A61K31/536;A61K31/5375;A61P1/04;A61P3/10;A61P5/14;A61P9/10;A61P11/06;A61P13/12;A61P17/00;A61P17/06;A61P19/08;A61P19/10;A61P21/04;A61P25/00;A61P25/02;A61P25/28;A61P29/00;A61P37/00;A61P37/02;A61P37/08;C07D205/04;C07D207/06;C07D207/14;C07D207/16;C07D211/58;C07D211/66;C07D309/14;C07D335/02;C07D401/04;C07D401/12;C07D403/06;C07D409/12;C07D413/00;C07D413/12;C07D417/00;C07D417/12;C07D451/04 |
主分类号 |
A61K31/535 |
代理机构 |
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代理人 |
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地址 |
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