发明名称 NOVEL SULFONYL DERIVATIVES
摘要 Sulfonyl derivatives represented by the following general formula (I): Q<1>-Q<2>-T<1>-Q<3>-SO2-Q<A> and drugs containing the same (wherein Q<1> is an optionally substituted, saturated or unsaturated, five- or six-membered cyclic hydrocarbon group, a five- or six-membered heterocyclic group, or the like; Q<2> is a single bond, oxygen, sulfur, C1-C6 alkylene or the like; Q<A> is optionally substituted arylalkenyl, heteroarylalkenyl or the like; and T<1> is carbonyl or the like). These compounds have potent FXa-inhibitory effects and promptly exert satisfactory and persistent antithrombotic effects through oral administration, thus being useful as anticoagulant agents little accompanied with side effects.
申请公布号 WO0009480(A1) 申请公布日期 2000.02.24
申请号 WO1999JP04344 申请日期 1999.08.11
申请人 DAIICHI PHARMACEUTICAL CO., LTD.;KOBAYASHI, SYOZO;KOMORIYA, SATOSHI;HAGINOYA, NORIYASU;SUZUKI, MASANORI;YOSHINO, TOSHIHARU;NAGAHARA, TAKAYASU;NAGATA, TSUTOMU;HORINO, HARUHIKO;ITO, MASAYUKI;MOCHIZUKI, AKIYOSHI 发明人 KOBAYASHI, SYOZO;KOMORIYA, SATOSHI;HAGINOYA, NORIYASU;SUZUKI, MASANORI;YOSHINO, TOSHIHARU;NAGAHARA, TAKAYASU;NAGATA, TSUTOMU;HORINO, HARUHIKO;ITO, MASAYUKI;MOCHIZUKI, AKIYOSHI
分类号 A61P7/02;C07D207/08;C07D207/12;C07D207/22;C07D211/34;C07D211/70;C07D213/56;C07D213/61;C07D213/73;C07D213/75;C07D213/82;C07D213/84;C07D213/89;C07D233/18;C07D233/54;C07D233/64;C07D233/88;C07D239/42;C07D239/48;C07D243/08;C07D277/28;C07D277/40;C07D401/04;C07D401/10;C07D401/12;C07D401/14;C07D405/04;C07D405/12;C07D409/04;C07D409/12;C07D409/14;C07D417/04;C07D417/12;C07D417/14;C07D491/048;(IPC1-7):C07D207/04;C07D295/22;C07D209/44;C07D333/68;C07D307/85;C07D495/04;C07D513/04;C07D498/04;C07D233/26;C07D217/26;C07D215/48;C07D235/08;C07D471/04;A61K31/44;A61K31/495;A61K31/55;A61K31/505;A61K31/535;A61K31/445;A61K31/53;A61K31/54;A61K31/435;A61K31/415;A61K31/47 主分类号 A61P7/02
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