发明名称 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1
摘要 The present invention relates to thiazolinones and also to pharmaceutical compositions comprising the compounds, as well as methods of use of the compounds for treatment of disorders associated with human 11-ß-hydroxysteroid dehydrogenase type 1 enzyme and for the preparation of a medicament which acts on the human 11- ß-hydroxysteroid dehydrogenase type 1 enzyme.
申请公布号 WO2007061661(A4) 申请公布日期 2009.01.29
申请号 WO2006US43951 申请日期 2006.11.13
申请人 AMGEN INC.;BIOVITRUM AB;HENRIKSSON, MARTIN;HOMAN, EVERT;JOHANSSON, LARS;VALLGARDA, JERK;WILLIAMS, MEREDITH;BERCOT, ERIC, A.;FOTSCH, CHRISTOPHER, H.;LI, AIWEN;CAI, GUOLIN;HUNGATE, RANDALL, W.;YUAN, CHESTER, CHENGUANG;TEGLEY, CHRISTOPHER;ST. JEAN, DAVID, J., JR.;HAN, NIANHE;HUANG, QI;LIU, QINGYIAN;BARTBEGER, MICHAEL, D.;MONIZ, GEORGE, A.;FRIZZLE, MATTHEW, J.;MARSHALL, TERESA, L. 发明人 HENRIKSSON, MARTIN;HOMAN, EVERT;JOHANSSON, LARS;VALLGARDA, JERK;WILLIAMS, MEREDITH;BERCOT, ERIC, A.;FOTSCH, CHRISTOPHER, H.;LI, AIWEN;CAI, GUOLIN;HUNGATE, RANDALL, W.;YUAN, CHESTER, CHENGUANG;TEGLEY, CHRISTOPHER;ST. JEAN, DAVID, J., JR.;HAN, NIANHE;HUANG, QI;LIU, QINGYIAN;BARTBEGER, MICHAEL, D.;MONIZ, GEORGE, A.;FRIZZLE, MATTHEW, J.;MARSHALL, TERESA, L.
分类号 C07D277/54;A61K31/426;A61K31/427;A61K31/428;A61P3/04;A61P3/06;A61P3/10;A61P9/12;A61P19/10;A61P25/24;C07D277/60;C07D417/04;C07D417/06;C07D417/12;C07D417/14 主分类号 C07D277/54
代理机构 代理人
主权项
地址