发明名称 CRYSTALLINE SALT FORM OF (S)-(2-(6-CHLORO-7-METHYL-1 H-BENZO[D]IMIDAZOL-2-YL)-2-METHYLPYRROLIDIN-1 -YL)(5-METHOXY-2-(2H-1,2,3-TRIAZOL-2-YL)PHENYL)METHANONE AS OREXIN RECEPTOR ANTAGONIST
摘要 The invention relates to a crystalline form of (S)-(2-(6-chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone hydrochloride, processes for the preparation thereof, pharmaceutical compositions containing said crystalline form, and its use as medicament, especially as orexin receptor antagonist.
申请公布号 SG11201604541W(A) 申请公布日期 2016.07.28
申请号 SG11201604541W 申请日期 2014.12.02
申请人 ACTELION PHARMACEUTICALS LTD 发明人 BOSS, CHRISTOPH;BROTSCHI, CHRISTINE;GUDE, MARKUS;HEIDMANN, BIBIA;SIFFERLEN, THIERRY;VON RAUMER, MARKUS;WILLIAMS, JODI T.
分类号 C07D403/14;A61K31/4192;A61P25/00 主分类号 C07D403/14
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