发明名称 |
EXTENDED RELEASE FORMULATION FOR OPTIMIZED DELIVERY OF AN HIV ATTACHMENT INHIBITOR |
摘要 |
A pharmaceutical composition contains the compound 1-benzoyl-4-[2-[4-methoxy-7-(3-methyl-1H-1,2,4-triazol-1--yl)-1-[(phosphonooxy)methyl]-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]-piperazine, and hydroxypropyl methyl cellulose (HPMC) having a viscosity of at least about 100 cP, wherein the composition does not contain any enzyme inhibitors. |
申请公布号 |
CA2735008(C) |
申请公布日期 |
2016.11.29 |
申请号 |
CA20092735008 |
申请日期 |
2009.09.03 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
BROWN, JONATHAN R.;TOALE, HELEN;DENNIS, ANDREW B.;TIMMINS, PETER |
分类号 |
A61K31/496;A61K31/00;A61P31/18 |
主分类号 |
A61K31/496 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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