发明名称 HETEROARYLOXY-BETA-CARBOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICINAL AGENTS
摘要 Heteroaryloxy-.beta.-carboline derivatives of general Formula I (I), wherein R1 is an optionally substituted heteroaryl residue, R2 is hydrogen, lower alkyl or lower alkoxyalkyl, X is a COOR3-group wherein R3 means H or lower alkyl, or represents a CONR4R5-group wherein R4 and R5 mean respectively hydrogen or lower alkyl, R4 and R5 being capable of forming, together with the nitrogen atom, a 5- -to 6-membered heterocycle, or means an oxadiazolyl residue of the formula or wherein R6 means hydrogen, lower alkyl or cycloalkyl, are valuable pharmaceuticals.
申请公布号 CA1315784(C) 申请公布日期 1993.04.06
申请号 CA19870531388 申请日期 1987.03.06
申请人 BIERE, HELMUT 发明人 BIERE, HELMUT;HUTH, ANDREAS;RAHTZ, DIETER;SCHMIECHEN, RALPH;SEIDELMANN, DIETER;STEPHENS, DAVID N.;ENGELSTOFT, MOGENS;HANSEN, JOHN B.
分类号 A61K31/435;A61K31/495;A61K31/505;A61P25/00;A61P25/08;A61P25/20;A61P25/28;C07D471/04 主分类号 A61K31/435
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