发明名称 CO-CRYSTAL OF CARFILZOMIB WITH MALEIC ACID AND PROCESS FOR THE PREPARATION OF PURE CARFILZOMIB
摘要 Aspects of the present application relates to co-crystal of carfilzomib with maleic acid, process for the preparation of co-crystal of carfilzomib with maleic acid, process for the preparation of pure carfilzomib from co-crystal of carfilzomib with maleic acid and process for the preparation of amorphous carfilzomib.
申请公布号 WO2016108204(A1) 申请公布日期 2016.07.07
申请号 WO2015IB60064 申请日期 2015.12.31
申请人 DR. REDDY'S LABORATORIES LIMITED 发明人 NADGOUD, RAMESH KUMAR;VASAM, SRIDHAR;MAKIREDDY, SIVA REDDY;MURKI, VEERENDER;GANORKAR, RAKESH;JOSE, JITHIN;PEDDI REDDY, SUBBA REDDY;CHAPPA, PRAVEEN
分类号 A61K47/48;C07C51/41 主分类号 A61K47/48
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