发明名称 |
TRIAZOLE-CONTAINING RELEASABLE LINKERS AND CONJUGATES COMPRISING THE SAME |
摘要 |
This invention relates to compounds comprising one or more therapeutic and/or diagnostic moieties and one or more functional moieties linked together via one or more triazole-containing linkers and to their intermediates and methods of their preparation. The triazole-containing linker may optionally contain one or more conditionally-cleavable or conditionally-transformable moieties and one or more spacer systems in between said moiety/moieties and the one or more therapeutic and/or diagnostic moieties. |
申请公布号 |
EP1909846(A2) |
申请公布日期 |
2008.04.16 |
申请号 |
EP20060783938 |
申请日期 |
2006.08.03 |
申请人 |
SYNTARGA B.V. |
发明人 |
BEUSKER, PATRICK HENRY;DE GROOT, FRANCISCUS MARINUS HENDRIKUS |
分类号 |
A61K47/48;A61P43/00;C07D249/04 |
主分类号 |
A61K47/48 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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