发明名称 AMINO-5-[SUBSTITUTED-4-(DIFLUOROMETHOXY)PHENYL]-5- PHENYLIMIDAZOLONE COMPOUNDS AS ß-SECRETASE INHIBITORS
摘要 <p>The present invention provides a 2-amino-5-[substituted-4-(difluoromethoxy)phenyl]-5-phenylimidazolone compound of formula (I) The present invention also provides methods for the use thereof to inhibit ß-secretase (BACE) and treat ß-amyloid deposits and neurofibrillary tangles.</p>
申请公布号 WO2008115552(A1) 申请公布日期 2008.09.25
申请号 WO2008US03681 申请日期 2008.03.20
申请人 WYETH;MALAMAS, MICHAEL SOTIRIOS;ROBICHAUD, ALBERT JEAN;PORTE, ALEXANDER MICHAEL;SOLVIBILE, WILLIAM RONALD;MORRIS, KOI MICHELE;ANTANE, SCHUYLER ADAM;KIM, JI-LN;MCDEVITT, ROBERT EMMETT 发明人 MALAMAS, MICHAEL SOTIRIOS;ROBICHAUD, ALBERT JEAN;PORTE, ALEXANDER MICHAEL;SOLVIBILE, WILLIAM RONALD;MORRIS, KOI MICHELE;ANTANE, SCHUYLER ADAM;KIM, JI-LN;MCDEVITT, ROBERT EMMETT
分类号 C07D233/88 主分类号 C07D233/88
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