发明名称 GLYCOSYLATED PRODRUGS, AND THEIR PROCESSES OF PREPARATION AND USE
摘要 Novel anthracycline prodrugs are provided herein of the Formula I below . (See formula I) In this formula, the various "R" groups have specifically-recited identity. These prodrugs have utility in combination with enzyme/tumour specific antibodies for use in cytostatic therapy.
申请公布号 CA2109304(A1) 申请公布日期 1992.10.31
申请号 CA19922109304 申请日期 1992.04.29
申请人 LABORATOIRES HOECHST;BEHRINGWERKE AG 发明人 JACQUESY, JEAN-CLAUDE;GESSON, JEAN-PIERRE;MONNERET, CLAUDE;MONDON, MARTINE;RENOUX, BRIGITTE;FLORENT, JEAN-CLAUDE;KOCH, MICHEL;TILLEQUIN, FRANCOIS;SEDLACEK, HANS H.;GERKEN, MANFRED;KOLAR, CENEK;GAUDEL, GILBERT;BOSSLET, KLAUS;CZECH, JOERG;HOFFMAN, DIETER;SEEMANN, GERHARD;SCHORLEMMER, HANS-ULRICH;DICKNEITE, GERHARD
分类号 A61K38/22;A61K31/70;A61K31/7028;A61K31/7034;A61K31/704;A61K38/46;A61K39/395;A61P35/00;A61P43/00;C07F7/18;C07H15/203;C07H15/252;C07H15/26;(IPC1-7):C07H15/252;C07F7/08;A61K47/42;A61K47/48 主分类号 A61K38/22
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