发明名称 3,7-DISUBSTITUTED INDOLE DERIVATIVE AND MEDICINAL COMPOSITION INCLUDING THE SAME
摘要 PROBLEM TO BE SOLVED: To provide a novel 3,7-disubstituted indole derivative that is useful as a medicine, particularly having theβ-adrenoreceptor stimulation action and a medicinal composition including the same. SOLUTION: The medicine is a 3,7-disubstituted indole derivative represented by the following formula [I] (wherein X is O, NH or S; Y is O, S or the like; R<1> is hydroxy, a lower alkoxy-carbonyl, a mono- or dialkylaminocarbonyl, carboxyl; R<2> and R<3> are each H, a lower alkyl; R<4> is H, phenyl, a heteroaryl or the like; R<5> is H, a halogen, hydroxy or the like; R<6> is H, a halogen, hydroxy, amino or the like; m is 0, 1 or 2; n is 1, 2, 3, 4 or 5; wherein R<4> is not H, when Y is O or SO2 ).
申请公布号 JP2003055344(A) 申请公布日期 2003.02.26
申请号 JP19990021483 申请日期 1999.01.29
申请人 DAINIPPON PHARMACEUT CO LTD 发明人 KATO SHIROU;HARADA HIROSHI;KINOSHITA IKUKO;KAWASHIMA KAZU
分类号 A61K31/00;A61K31/40;A61K31/403;A61K31/404;A61K31/4045;A61P3/00;A61P3/04;A61P3/10;A61P43/00;C07D209/16;(IPC1-7):C07D209/16 主分类号 A61K31/00
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