摘要 |
<p>Cpds. of formula (I): (where R1 is H, halogen, lower alkyl or NO2 (pref. 7-Cl 7-NO2); R2 is H, lower alkyl or di(lower alkyl)amino-lower alkyl (pref. H, Me or 2-diethylaminoethyl); R3 is pyridyl phenyl or halophenyl (pref. Ph, 2-pyridyl or 2-fluoro- or 2-chlorophenyl); B is CO or CH2) prepd. by treating a cpd. (II); with a reducing agent, pref. HI (esp. formed in situ) or NH2OH. Cpds. (I) are sedatives, tranquillisers, anticonvulsants and muscle relaxants.</p> |