发明名称 |
POLYMORPH FORMS OF PYRROLIDINE-2,5-DIONE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF |
摘要 |
Two distinct crystalline forms of a 3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione are provided. The compound 3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione is an IDO1 inhibitor. The crystalline forms may be used in the preparation of pharmaceutical compositions. |
申请公布号 |
CA2929837(A1) |
申请公布日期 |
2016.11.14 |
申请号 |
CA20162929837 |
申请日期 |
2016.05.12 |
申请人 |
PFIZER INC.;ITEOS THERAPEUTICS |
发明人 |
CAUWENBERGHS, SANDRA;CROSIGNANI, STEFANO;DRIESSENS, GREGORY;KEENE, NANDELL;FICHTNER, MICHAEL W. |
分类号 |
C07D403/04;A61K31/404 |
主分类号 |
C07D403/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|