发明名称 POLYMORPH FORMS OF PYRROLIDINE-2,5-DIONE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF
摘要 Two distinct crystalline forms of a 3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione are provided. The compound 3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione is an IDO1 inhibitor. The crystalline forms may be used in the preparation of pharmaceutical compositions.
申请公布号 CA2929837(A1) 申请公布日期 2016.11.14
申请号 CA20162929837 申请日期 2016.05.12
申请人 PFIZER INC.;ITEOS THERAPEUTICS 发明人 CAUWENBERGHS, SANDRA;CROSIGNANI, STEFANO;DRIESSENS, GREGORY;KEENE, NANDELL;FICHTNER, MICHAEL W.
分类号 C07D403/04;A61K31/404 主分类号 C07D403/04
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