发明名称 |
Pyridylalkyl imidazole-2-thiols |
摘要 |
Potent dopamine- beta -hydroxylase inhibitors having the formula: <IMAGE> which are useful to inhibit dopamine- beta -hydroxylase activity, pharmaceutical compositions including these inhibitors, and methods of using these inhibitors to inhibit dopamine- beta -hydroxylase activity in mammals. Also disclosed are novel intermediates useful in preparing the presently invented inhibitors.
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申请公布号 |
US4634711(A) |
申请公布日期 |
1987.01.06 |
申请号 |
US19850761936 |
申请日期 |
1985.08.02 |
申请人 |
SMITHKLINE BECKMAN CORPORATION |
发明人 |
KAISER, CARL;KRUSE, LAWRENCE I.;ROSS, STEPHEN T. |
分类号 |
A61K31/44;A61K31/4412;A61K31/4418;A61K31/4427;A61P1/04;A61P7/10;A61P9/04;A61P9/08;A61P9/12;A61P25/02;A61P43/00;C07D213/64;C07D213/65;C07D213/89;C07D401/06;C12N9/99;(IPC1-7):A61K31/415 |
主分类号 |
A61K31/44 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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