发明名称 OPTICALLY ACTIVE AZETIDINONES AND PROCESS FOR PRODUCTION THEREOF
摘要 <p>Compounds of formula (I), wherein Y represents an acetyl, 1-hydroxyethyl or 1-fluoroethyl group, R1 represents a hydrogen atom or an easily splittable amino-protecting group, and R2 and R3 are identical or different and each represents a hydrogen atom, a lower alkyl group, a phenyl group, a benzyl group or a diphenylmethyl group, or R2 and R3 together represent a lower alkylene group; and processes for production thereof. These compounds are useful as synthesis intermediates for production of various medicines, particularly carbapenam or carbapenem antibiotics, such as a carbapenem antibiotic of formula (A) which has excellent antimicrobial activity and relatively good stability to kidney dehydropeptidase.</p>
申请公布号 WO8804656(A1) 申请公布日期 1988.06.30
申请号 WO1987JP00991 申请日期 1987.12.18
申请人 SANRAKU INCORPORATED 发明人 YOSHIOKA, TAKEO;WATANABE, MACHIKO;FUKAGAWA, YASUO;ISHIKURA, TOMOYUKI
分类号 C07D405/06;C07D205/08;C07D405/04;C07D521/00;(IPC1-7):C07D405/04 主分类号 C07D405/06
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