COMPOUNDS FOR AND METHOD OF INHIBITING PHOSPHODIESTERASE IV
摘要
Novel compounds which are effective PDE IV inhibitors are disclosed. The compounds possess similar or improved PDE IV inhibition as compared to rolipram, with improved selectivity with regard to, e.g., PDE III inhibition. Preferred compounds are 3-(3-cyclopentyloxy-4-methoxy-benzylamino)-4-hydroxymethyl pyrazole and 3-(3-cyclopentyloxy-4-methoxybenzylamino)-4-methoxymethylpyrazole.
申请公布号
WO9600218(A1)
申请公布日期
1996.01.04
申请号
WO1995US08981
申请日期
1995.06.23
申请人
EURO-CELTIQUE, S.A.;CAVALLA, DAVID;CHASIN, MARK;DOLBY, LLOYD;FRITH, RICHARD, W.
发明人
CAVALLA, DAVID;CHASIN, MARK;DOLBY, LLOYD;FRITH, RICHARD, W.