发明名称 |
5-FLUORO-4-IMINO-3-(ALKYL/SUBSTITUTED ALKYL)-1-(ARYLSULFONYL)-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE AND PROCESSES FOR THEIR PREPARATION |
摘要 |
Provided herein are 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1H)-one and processes for their preparation which may include the use of an alkali carbonate and an alkylating agent; |
申请公布号 |
US2016280662(A1) |
申请公布日期 |
2016.09.29 |
申请号 |
US201615173493 |
申请日期 |
2016.06.03 |
申请人 |
Adama Makhteshim Ltd. |
发明人 |
Choy Nakyen;Ross, JR. Ronald |
分类号 |
C07D239/47 |
主分类号 |
C07D239/47 |
代理机构 |
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代理人 |
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主权项 |
1. A method of making compounds of Formula III, including the steps of contacting a compound of Formula II with an alkali carbonate and an alkylating agent, and forming a compound of Formula III: wherein R1 is selected from the group consisting of: and R2 is selected from the group consisting of: |
地址 |
Airport City IL |