发明名称 |
ANALOGUES OF BESTATIN |
摘要 |
<p>Bestatin, which is (2S,3R)-3-amino-2-hydroxy-4-phenylbutanoyl!-L-leucine, and related compounds which inhibit aminopeptidase B, leucino aminopeptidase and Bleomycin hydrolase, enhance the antitumor effect of Bleomycin and exhibit an antifertility effect were synthesized and tested.</p> |
申请公布号 |
CA1104156(A) |
申请公布日期 |
1981.06.30 |
申请号 |
CA19760257393 |
申请日期 |
1976.07.20 |
申请人 |
MICROBIAL CHEM RES FOUND |
发明人 |
UMEZAWA, HAMAO;AOYAGI, TAKAAKI;TAKITA, TOMOHISA;NISHIZAWA, RINZO;SAINO, TETSUSHI |
分类号 |
A61K31/195;A61K38/00;A61P43/00;C07C67/00;C07C227/00;C07C229/22;C07C229/34;C07C231/00;C07C231/02;C07C231/06;C07C231/12;C07C237/12;C07C237/14;C07C237/20;C07C239/00;C07C271/22;C07C313/00;C07C323/59;C07K5/02;C07K5/06;(IPC1-7):C07C103/52 |
主分类号 |
A61K31/195 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|