发明名称 Process for preparing substituted 5-fluoro-1H-pyrazolopyridines
摘要 The present application relates to a novel and efficient process for preparing novel substituted 5-fluoro-1H-pyrazolopyridines of the formula (VI); which are suitable as an intermediate for production of medicaments and for production of medicaments for treatment and/or prophylaxis of cardiovascular disorders. More particularly, the 5-fluoro-1H-pyrazolopyridines of the formula (VI) are suitable for preparation of the compound of the formula (I) ; which serves for production of medicaments, for production of medicaments for treatment and/or prophylaxis of cardiovascular disorders.
申请公布号 US9604948(B2) 申请公布日期 2017.03.28
申请号 US201514796703 申请日期 2015.07.10
申请人 ADVERIO PHARMA GMBH 发明人 Fey Peter;Grunenberg Alfons;Bierer Donald
分类号 A01N43/54;C07D295/104;C07D265/30;C07D471/04;C07C309/04;C07C317/04;C07D295/067;C07C303/28 主分类号 A01N43/54
代理机构 Buchanan Ingersoll & Rooney PC 代理人 Buchanan Ingersoll & Rooney PC
主权项 1. A compound of formula (I) in crystalline form of polymorph Iwherein the x-ray diffractogram of the compound exhibits peak maxima of the 2 theta angle at 5.9, 6.9, 22.7.
地址 Schoenefeld DE