发明名称 |
Process for preparing substituted 5-fluoro-1H-pyrazolopyridines |
摘要 |
The present application relates to a novel and efficient process for preparing novel substituted 5-fluoro-1H-pyrazolopyridines of the formula (VI);
which are suitable as an intermediate for production of medicaments and for production of medicaments for treatment and/or prophylaxis of cardiovascular disorders. More particularly, the 5-fluoro-1H-pyrazolopyridines of the formula (VI) are suitable for preparation of the compound of the formula (I)
;
which serves for production of medicaments, for production of medicaments for treatment and/or prophylaxis of cardiovascular disorders. |
申请公布号 |
US9604948(B2) |
申请公布日期 |
2017.03.28 |
申请号 |
US201514796703 |
申请日期 |
2015.07.10 |
申请人 |
ADVERIO PHARMA GMBH |
发明人 |
Fey Peter;Grunenberg Alfons;Bierer Donald |
分类号 |
A01N43/54;C07D295/104;C07D265/30;C07D471/04;C07C309/04;C07C317/04;C07D295/067;C07C303/28 |
主分类号 |
A01N43/54 |
代理机构 |
Buchanan Ingersoll & Rooney PC |
代理人 |
Buchanan Ingersoll & Rooney PC |
主权项 |
1. A compound of formula (I) in crystalline form of polymorph Iwherein the x-ray diffractogram of the compound exhibits peak maxima of the 2 theta angle at 5.9, 6.9, 22.7. |
地址 |
Schoenefeld DE |