发明名称 |
SYDNONE DERIVATIVES FOR CONJUGATION OF COMPOUNDS OF INTEREST |
摘要 |
The present invention relates to a process for the preparation of a first compound of interest C1 functionalized with a sydnone compound and to the corresponding functionalized C1 compound of interest. The present invention also relates to a process for the preparation of a conjugate of two compounds of interest C1 and C2 implying a sydnone compound and to the obtained conjugate. The present invention also relates to a process for preparing a compound of interest C2 comprising a strained alkyne moiety functionalized with a sydnone and to the corresponding functionalized compound of interest C2. It also relates to novel sydnone compounds substituted in position 4, which may be used in the above processes. |
申请公布号 |
US2017081300(A1) |
申请公布日期 |
2017.03.23 |
申请号 |
US201515310459 |
申请日期 |
2015.05.15 |
申请人 |
UNIVERSITE DE STRASBOURG ;CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE ;COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES |
发明人 |
TARAN FREDERIC;WAGNER ALAIN;KOLODYCH SERGII;KONIEV OLEKSANDR |
分类号 |
C07D271/04;C07D495/04;C07D231/54;C07K16/00;C07K14/765 |
主分类号 |
C07D271/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
STRASBOURG FR |