发明名称 |
CHIRAL REAGENTS FOR PREPARATION OF HOMOGENEOUS OLIGOMERS |
摘要 |
We provide diastereomerically pure or substantially diastereomerically pure activated phosphoramidochloridate morpholino nucleosides, methods of their preparation, and methods of their use in stereospecific coupling for stereospecific synthesis of diastereomerically pure phosphorodiamidate morpholino oligomers (PMOs). |
申请公布号 |
WO2017024264(A2) |
申请公布日期 |
2017.02.09 |
申请号 |
WO2016US45876 |
申请日期 |
2016.08.05 |
申请人 |
EISAI R&D MANAGEMENT CO., LTD. |
发明人 |
ENDO, Atsushi;YU, Robert T.;FANG, Francis;CHOI, Hyeong Wook;SHAN, Mingde |
分类号 |
C07F9/6558;A61K31/713;C07F9/6561;C07H21/00 |
主分类号 |
C07F9/6558 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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