发明名称 ACYCLIC CYANOETHYLPYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS
摘要 The instant invention provides compounds of formula I which are JAK inhibitors, and as such are useful for the treatment of JAK-mediated diseases such as rheumatoid arthritis, asthma, COPD and cancer.
申请公布号 EP2976341(A4) 申请公布日期 2016.10.12
申请号 EP20140770056 申请日期 2014.03.19
申请人 MERCK SHARP & DOHME CORP. 发明人 DINSMORE, CHRISTOPHER;FULLER, PETER;GUERIN, DAVID;KATZ, JASON DAVID;THOMPSON, CHRISTOPHER F.;FALCONE, DANIELLE;DENG, WEI;TORRES, LUIS;ZENG, HONGBO;BAI, YUNFENG;FU, JIANMIN;KONG, NORMAN;LIU, YUMEI;ZHENG, ZHIXIANG;SCOTT, MARK E.
分类号 C07D471/04;A61K31/437;A61K31/4375;A61P25/00;A61P35/00;A61P37/00;C07D487/04;C07D487/08;C07D487/14 主分类号 C07D471/04
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