发明名称 |
HETERO-CONDENSED RING COMPOUND |
摘要 |
A compound represented by the formula (I) or a salt thereof:
wherein a ring Z is a 5 to 6-membered heteroaromatic ring having one or two heteroatoms in the ring; X 1 is a hydrogen atom, a hydroxy group, a hydroxy C 1-6 alkyl group, -B(OH) 2 , a boronate ester group, a cyclic boronate ester group, a boranyl group, a cyclic boranyl group, -BF 3 M n1 , -Sn(R 12 )(R 13 )(R 14 ), a leaving group, a carboxy group, a formyl group, or -NR 16 R 17 ; and X 2 is a hydrogen atom or -CO 2 R 18 . |
申请公布号 |
EP3026054(A1) |
申请公布日期 |
2016.06.01 |
申请号 |
EP20140829168 |
申请日期 |
2014.07.18 |
申请人 |
EISAI R&D MANAGEMENT CO., LTD. |
发明人 |
TANAKA, KEIGO;FUKUYAMA, TAKASHI;MURAI, NORIO;ITANO, WATARU;HIROTA, SHINSUKE;IIDA, DAISUKE;AZUMA, HIROSHI |
分类号 |
C07D491/048;A61K31/34;A61K31/381;A61K31/407;A61K31/429;A61K31/4355;A61K31/4985;A61K31/5025;A61K31/519;A61P1/04;A61P9/10;A61P31/10;C07B61/00;C07D493/04;C07D495/04;C07D513/04;C07F5/02;C07F7/22 |
主分类号 |
C07D491/048 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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