发明名称 |
4-(8-METHOXY-1-((1-METHOXYPROPAN-2-YL)-2-(TETRAHYDRO-2H-PYRAN-4-YL)-1H-IMIDAZO[4,5-c]QUINOLIN-7-YL)-3,5-DIMETHYLISOXAZOLE AND ITS USE AS BROMODOMAIN INHIBITOR |
摘要 |
Novel quinoline compounds of formula (I), pharmaceutical compositions containing such compounds and their use in therapy, as bromodomain inhibitors. |
申请公布号 |
EA023374(B1) |
申请公布日期 |
2016.05.31 |
申请号 |
EA20140090200 |
申请日期 |
2012.08.15 |
申请人 |
GLAXOSMITHKLINE LLC |
发明人 |
DEMONT EMMANUEL, HUBERT;JONES KATHERINE, LOUISE;WATSON ROBERT, J. |
分类号 |
C07D471/04;A61K31/4745;A61P29/00;A61P37/00 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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