发明名称 CO-CRYSTALS OF (S)-N-METHYL-8-(1-((2'-METHYL-[4,5'-BIPYRIMIDIN]-6-YL)AMINO)PROPAN-2-YL)QUINOLINE-4-CARBOXAMIDE AND DEUTERATED DERIVATIVES THEREOF AS DNA-PK INHIBITORS
摘要 wherein each of R1 and R2 is H or 2H and a co-crystal former selected from adipic acid, citric acid, fumaric acid, maleic acid, succinic acid, or benzoic acid. Also within the scope of this invention are methods of making and using the same.
申请公布号 SG11201602962P(A) 申请公布日期 2016.05.30
申请号 SG11201602962P 申请日期 2014.10.17
申请人 VERTEX PHARMACEUTICALS INCORPORATED 发明人 NTI-ADDAE, KWAME, WIREDU;O'NEIL, SIMON, ADAM;ZHANG, YUEGANG;WALDO, MICHAEL;MUDUNURI, PRAVEEN;SONG, BIN;VAN ALSTEN, JOHN GREGG;STROHMEIER, MARK;STAVROPOULOS, KATHY;KADIYALA, IRINA NIKOLAEVNA;NAVAMAL, METTACHIT
分类号 C07D401/14;A61K31/506;A61P35/00 主分类号 C07D401/14
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