发明名称 Preparation method for pyrrolidine-2-carboxylic acid derivatives
摘要 The present invention relates to the field of medical synthesis, in particular to a preparation method for pyrrolidine-2-carboxylic acid derivatives. The present invention adopts the following technical solution: providing a compound having a structure of formula (E), wherein R is R1 or R2, R1 is C1-C6 an alkyl, benzyl, p-methoxybenzyl, or p-nitrobenzyl group, and R2 is hydrogen; R3 is a protecting group of the carboxyl group; and P1 is a protecting group on nitrogen.;
申请公布号 US2016145208(A1) 申请公布日期 2016.05.26
申请号 US201414898465 申请日期 2014.06.23
申请人 ZHEJIANG JIUZHOU PHARMACEUTICAL CO., LTD. 发明人 ZHANG Bin;LI Yuanqiang;CHE Daqing;QIAN Lingfeng;ZHU Guoliang;YE Wenfa
分类号 C07D207/22 主分类号 C07D207/22
代理机构 代理人
主权项 1. A compound of formula E, wherein R is R1 or R2, R1 is C1˜C6 alkyl, benzyl, p-methoxybenzyl or p-nitrobenzyl, R2 is a hydrogen atom; R3 is a protecting group for carboxyl; P1 is a protecting group of nitrogen.
地址 Zhejiang CN