发明名称 |
ANDROGEN RECEPTOR MODULATORS AND THEIR USE AS ANTI-CANCER AGENTS |
摘要 |
Compounds having therapeutic potential as androgen receptor modulators and anti- cancer agents, and methods of making such compounds, are provided. The compounds are structurally related to bicalutamide, enobosarm and enzalutamide, but bear a 3,5-bis- CF3 group as a substituent. |
申请公布号 |
WO2016079521(A1) |
申请公布日期 |
2016.05.26 |
申请号 |
WO2015GB53527 |
申请日期 |
2015.11.19 |
申请人 |
UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED |
发明人 |
WESTWELL, ANDREW D;PERTUSATI, FABRIZIO;MCGUIGAN, CHRISTOPHER;BRANCALE, ANDREA;BASSETTO, MARCELLA;FERLA, SALVATORE;KANDIL, SAHAR |
分类号 |
C07D233/86;A61K31/4166;A61P35/00;C07C233/01 |
主分类号 |
C07D233/86 |
代理机构 |
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代理人 |
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地址 |
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