| 摘要 |
The present invention relates to compounds of formula (I) and to salts thereof, wherein R1, R2, and Q have any of the values defined in the specification, and compositions and uses thereof. The compounds are useful as inhibitors of bromodomains. Also included are pharmaceutical compositions comprising a compound of formula (I) or a pharmaceutically acceptable salt thereof, and methods of using such compounds and salts in the treatment of various bromodomain-mediated disorders. |
| 申请人 |
GENENTECH, INC.;CONSTELLATION PHARMACEUTICALS, INC. |
发明人 |
ALBRECHT, BRIAN, K.;BELLON, STEVEN, F.;BURDICK, DANIEL, J.;COTE, ALEXANDRE;CRAWFORD, TERRY;DAKIN, LES, A.;HEWITT, MICHAEL, CHARLES;HSIAO-WEI TSUI, VICKIE;LEBLANC, YVES;MAGNUSON, STEVEN, R.;NASVESCHUK, CHRISTOPHER, G.;ROMERO, F. ANTHONY;TANG, YONG;TAYLOR, ALEXANDER, M.;WANG, SHUMEI |
