发明名称 Processes for producing cycloalkylcarboxamido-pyridine benzoic acids
摘要 The present invention relates to presses for preparing Cystic Fibrosis transmembrane conductance regulator (CFTR) correctors such as the compound 3-(6-( (2,2difliuorobenzo [d] [1.3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin 2-yl)benzoic acid (Compound 1) in substantially free form useful in the treatment of cystic fibrosis, F O N N N CO 2 H Compound 1.
申请公布号 AU2013205160(B2) 申请公布日期 2016.05.19
申请号 AU20130205160 申请日期 2013.04.14
申请人 VERTEX PHARMACEUTICALS INCORPORATED 发明人 SIESEL, DAVID
分类号 C07D213/73;C07D405/12 主分类号 C07D213/73
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