发明名称 |
PRODUCING METHOD OF F-18-LABELED AMYLOID BETA LIGAND |
摘要 |
PROBLEM TO BE SOLVED: To provide a producing method making rigid and safe production of F-18-labeled tracer possible.SOLUTION: A [F-18] fluoro-pegylated (aryl/heteroaryl vinyl)-phenylmethyl amine derivative shown by a formula 1 is produced by performing a radiolabeled (aryl/heteroaryl vinyl)-phenylmethyl amine derivative having a halogen-group or a sulfonyl oxy group with F-18 fluorinating agent. The X is CH or N. The n is 1-6.SELECTED DRAWING: None |
申请公布号 |
JP2016047831(A) |
申请公布日期 |
2016.04.07 |
申请号 |
JP20150208782 |
申请日期 |
2015.10.23 |
申请人 |
PIRAMAL IMAGING SA |
发明人 |
MATHIAS BERNDT;MATTHIAS FRIEBE;FABRICE SAMSON;RAINER BRAUN;GUNNAR GARKE;MARIANNE PATT;ANDREAS SCHILDAN;CHRISTOPH SMUDA |
分类号 |
C07C213/08;A61K9/08;A61K47/04;A61K47/10;A61K47/22;A61K51/00;C07C217/80;C07D213/64 |
主分类号 |
C07C213/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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