发明名称 PRODUCING METHOD OF F-18-LABELED AMYLOID BETA LIGAND
摘要 PROBLEM TO BE SOLVED: To provide a producing method making rigid and safe production of F-18-labeled tracer possible.SOLUTION: A [F-18] fluoro-pegylated (aryl/heteroaryl vinyl)-phenylmethyl amine derivative shown by a formula 1 is produced by performing a radiolabeled (aryl/heteroaryl vinyl)-phenylmethyl amine derivative having a halogen-group or a sulfonyl oxy group with F-18 fluorinating agent. The X is CH or N. The n is 1-6.SELECTED DRAWING: None
申请公布号 JP2016047831(A) 申请公布日期 2016.04.07
申请号 JP20150208782 申请日期 2015.10.23
申请人 PIRAMAL IMAGING SA 发明人 MATHIAS BERNDT;MATTHIAS FRIEBE;FABRICE SAMSON;RAINER BRAUN;GUNNAR GARKE;MARIANNE PATT;ANDREAS SCHILDAN;CHRISTOPH SMUDA
分类号 C07C213/08;A61K9/08;A61K47/04;A61K47/10;A61K47/22;A61K51/00;C07C217/80;C07D213/64 主分类号 C07C213/08
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