发明名称 PYRROLCARBOXAMIDE DERIVATIVES FOR THE INHBITION OF ERK5
摘要 The invention provides compounds of formula (I) or a tautomer, stereoisomer, N-oxide, pharmaceutically acceptable salt or solvate thereof. The compounds are useful for the prophylaxis or treatment of a disease state or condition mediated by ERK5, in particular cancers.
申请公布号 WO2016042341(A1) 申请公布日期 2016.03.24
申请号 WO2015GB52707 申请日期 2015.09.18
申请人 CANCER RESEARCH TECHNOLOGY LIMITED 发明人 REUILLON, TRISTAN;MILLER, DUNCAN;MYERS, STEPHANIE;MOLYNEUX, LAUREN;CANO, CELINE;HARDCASTLE, IAN;RIGOREAU, LAURENT;GOLDING, BERNARD;NOBLE, MARTIN;GRIFFIN, ROGER
分类号 C07D403/12;A61K31/506;A61P35/00;C07D401/12;C07D401/14;C07D403/14;C07D405/14;C07D413/12;C07D413/14 主分类号 C07D403/12
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