TEDIZOLID PHOSPHATE, INTERMEDIATE AND PREPARATION METHOD THEREOF

摘要

Provided is a preparation method for tedizolid phosphate, an intermediate thereof of formula VII and a preparation method for the intermediates of formulae V, VII, IX and X. The preparation method has a short route, mild reaction conditions and is green and environmentally friendly. Dibenzyl diisopropylamino phosphite is used as a phosphorylation agent, avoiding the production of dimeric products and enabling a higher yield of the preparation method.