发明名称 テトラゾール化合物の脱保護方法
摘要 The present invention relates to a method of deprotecting a tetrazole compound, useful as an intermediate for angiotensin II receptor blockers, and provides a novel production method of angiotensin II receptor blockers. Provided is a production method of a compound represented by the formula [3] or [4] or a salt thereof, including (i) reducing a compound represented by the formula [1] or [2] or a salt thereof in the presence of a metal catalyst and an alkaline earth metal salt, or (ii) reacting the compound with a particular amount of Brønsted acid: wherein each symbol is as defined in the present specification.
申请公布号 JP5881837(B2) 申请公布日期 2016.03.09
申请号 JP20140538604 申请日期 2013.09.26
申请人 株式会社エーピーアイ コーポレーション 发明人 関 雅彦
分类号 C07D257/04;B01J27/053;B01J27/185;C07D403/10;C07D405/14 主分类号 C07D257/04
代理机构 代理人
主权项
地址