发明名称 NOVEL FORMULATIONS OF A BRUTON'S TYROSINE KINASE INHIBITOR
摘要 Described herein is the Brutons tyrosine kinase (Btk) inhibitor 1-((R)-3-(4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one, including novel pharmaceutical formulations thereof. Also disclosed are pharmaceutical compositions that include the Btk inhibitor, as well as methods of using the Btk inhibitor, alone or in combination with other therapeutic agents, for the treatment of autoimmune diseases or conditions, heteroimmune diseases or conditions, cancer, including lymphoma, and inflammatory diseases or conditions.
申请公布号 CA2955747(A1) 申请公布日期 2016.02.11
申请号 CA20152955747 申请日期 2015.08.07
申请人 PHARMACYCLICS LLC 发明人 TAY, PEARL SHWE-CHO;MINIKIS, RYAN MITCHELL;HULVAT, JAMES FRANCIS;MCVEY, ALEXANDER JACOB;SHU, CASSANDRA;ATLURI, HARISHA;KUEHL, ROBERT;CHONG, CHING WAH
分类号 A61K31/519;A61K9/26;C07D487/04 主分类号 A61K31/519
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