发明名称 |
NOVEL FORMULATIONS OF A BRUTON'S TYROSINE KINASE INHIBITOR |
摘要 |
Described herein is the Brutons tyrosine kinase (Btk) inhibitor 1-((R)-3-(4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one, including novel pharmaceutical formulations thereof. Also disclosed are pharmaceutical compositions that include the Btk inhibitor, as well as methods of using the Btk inhibitor, alone or in combination with other therapeutic agents, for the treatment of autoimmune diseases or conditions, heteroimmune diseases or conditions, cancer, including lymphoma, and inflammatory diseases or conditions. |
申请公布号 |
CA2955747(A1) |
申请公布日期 |
2016.02.11 |
申请号 |
CA20152955747 |
申请日期 |
2015.08.07 |
申请人 |
PHARMACYCLICS LLC |
发明人 |
TAY, PEARL SHWE-CHO;MINIKIS, RYAN MITCHELL;HULVAT, JAMES FRANCIS;MCVEY, ALEXANDER JACOB;SHU, CASSANDRA;ATLURI, HARISHA;KUEHL, ROBERT;CHONG, CHING WAH |
分类号 |
A61K31/519;A61K9/26;C07D487/04 |
主分类号 |
A61K31/519 |
代理机构 |
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地址 |
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