发明名称 |
COFORMER SALTS OF (2S,3S)-METHYL 7-FLUORO-2-(4-FLUOROPHENYL)-3-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-4-OXO-1,2,3,4-TETRAHYDROQUINOLINE-5-CARBOXYLATE AND METHODS OF PREPARING THEM |
摘要 |
Described herein are coformer salts of (2S,3S)-methyl 7-fluoro-2-(4-fluorophenyl)-3- ( 1-methyl- 1H- 1,2,4-triazol-5-yl)-4-oxo-l,2,3,4-tetrahydroquinoline-5-carboxylate optionally as a solvate and additionally optionally as a hydrate, including crystalline forms, and methods of preparing the (2S,3S)-methyl 7-fluoro-2-(4-fluorophenyl)-3-( 1-methyl- 1H-1, 2,4-triazol-5- yl)-4-oxo-l,2,3,4-tetrahydroquinoline-5-carboxylate optionally as a coformer salts. |
申请公布号 |
CA2956714(A1) |
申请公布日期 |
2016.02.04 |
申请号 |
CA20152956714 |
申请日期 |
2015.07.30 |
申请人 |
MEDIVATION TECHNOLOGIES, INC. |
发明人 |
HENDERSON, MARK;CAMPBELL, COLM;JAGUSCH, CARSTEN;HERZ, CHRISTIAN KLAUS;BAUER, NICO;BONNAUD, THIERRY;LAMBERT, OLIVIER |
分类号 |
C07D215/22;C07D221/04 |
主分类号 |
C07D215/22 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|