发明名称 |
Methods for the preparation of 5-[2-[7-(trifluoromethyl)-5-[4-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]ethynyl]-2-pyridinamine |
摘要 |
The present disclosure provides methods for preparing 5-[2-[7-(trifluoromethyl)-5-[4(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]ethynyl]-2-pyridinamine (compound A), which is useful for the treatment of depression and other CNS disorders. The present methods are useful for preparing compound A on large scale in manufacturing facilities. |
申请公布号 |
NZ621156(A) |
申请公布日期 |
2016.01.29 |
申请号 |
NZ20120621156 |
申请日期 |
2012.10.01 |
申请人 |
F. HOFFMANN-LA ROCHE AG |
发明人 |
WICHMANN JUERGEN;WOLTERING THOMAS;YANG JASON;BAILEY DANIEL;SRIVASTAVA AMIT;MILLER DOREEN;BACHMANN STEPHAN;BRICE JODIE;CEDILOTE MIALL;DONG ZHIMING;HILDBRAND STEFAN;SPURR PAUL;ZHANG PINGSHENG |
分类号 |
C07D487/04;A61K31/4162;A61K31/519;C07D213/73 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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