发明名称 Prodrugs of gaba analogs, compositions and uses thereof
摘要 The present invention provides prodrugs of GABA analogs, pharmaceutical compositions of prodrugs of GABA analogs and methods for making prodrugs of GABA analogs. The present invention also provides methods for using prodrugs of GABA analogs and methods for using pharmaceutical compositions of prodrugs of GABA analogs for treating or preventing common diseases and/or disorders.
申请公布号 US9238616(B2) 申请公布日期 2016.01.19
申请号 US201514792243 申请日期 2015.07.06
申请人 XenoPort, Inc. 发明人 Gallop Mark A.
分类号 A61K31/27;A61K31/24;C07C229/28;C07C309/29;A61K31/22 主分类号 A61K31/27
代理机构 Polsinelli PC 代理人 Polsinelli PC
主权项 1. A compound of Formula (I): or a pharmaceutically acceptable salt thereof, wherein X is oxygen; n is 0; each of R1, R3, R6 and R7 is hydrogen; Y is oxygen; and R4 and R5, together with the carbon atom to which they are attached, form a C7-cycloalkenyl ring that is substituted with an ethanyl moiety.
地址 Santa Clara CA US