发明名称 CRYSTALLINE SULFATE SALT FORMS OF AN 8-AZABICYCLO[3.2.1]OCTANE COMPOUND
摘要 The invention provides a crystalline sulfate salt of 3-endo-(8-{2-[cyclohexylmethyl-((S)-2,3-dihydroxy-propionyl)amino]ethyl}-8-aza-bicyclo[3.2.1]oct-3-yl)benzamide or a solvate thereof. The invention also provides pharmaceutical compositions comprising such crystalline salt forms, methods of using such crystalline salt forms to treat diseases associated with mu opioid receptor activity, and processes useful for preparing such crystalline salt forms.
申请公布号 CA2678073(C) 申请公布日期 2016.01.05
申请号 CA20082678073 申请日期 2008.02.27
申请人 THERAVANCE, INC. 发明人 DALZIEL, SEAN;PREZA, LETICIA M.;RAPTA, MIROSLAV;COLSON, PIERRE-JEAN
分类号 C07D451/02;A61K31/46 主分类号 C07D451/02
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