发明名称 |
AN ORGANOCATALYTIC ASYMMETRIC SYNTHESIS OF ANTIDEPRESSANTS |
摘要 |
The present invention relates to a short enantioselective synthesis of 1-amino aryl tetraline compounds of Formula 1 via nucleophilic enamine catalysis using organocatalyst such as proline. wherein R1 and R2 represent independent of each other hydrogen, (un)substituted or substituted amine; R3 and R4 represent independent of each other hydrogen or halogen. |
申请公布号 |
WO2015193921(A1) |
申请公布日期 |
2015.12.23 |
申请号 |
WO2015IN50048 |
申请日期 |
2015.06.22 |
申请人 |
COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH |
发明人 |
VAITHIYANATHAN, VENKATARAMASUBRAMANIAN;KALSHETTI, RUPALI GUNDAPPA;ARUMUGAM, SUDALAI |
分类号 |
C07C249/02;C07C251/20 |
主分类号 |
C07C249/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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