发明名称 |
SOLID FORMS OF AN ANTIVIRAL COMPOUND |
摘要 |
Crystalline solid forms of methyl {(2S)-1-[(2S,5S)-2-(9-{2-[(2S,4S)-1-{(2R)-2- [(methoxycarbonyl)amino] -2-phenylacetyl} -4-(methoxymethyl)pyrrolidin-2-yl] - 1 H-imidazol-5 - yl} -1, 11 -dihydroisochromeno[4',3':6,7]naphtho[ 1,2-d]imidazol-2-yl)-5-methylpyrrolidin- 1 -yl]-3- methyl-l-oxobutan-2-yl} carbamate (Compound I) were prepared and characterized in the solid state: Also provided are processes of manufacture and methods of using these crystalline forms. |
申请公布号 |
CA2951188(A1) |
申请公布日期 |
2015.12.17 |
申请号 |
CA20152951188 |
申请日期 |
2015.06.08 |
申请人 |
GILEAD PHARMASSET LLC |
发明人 |
LAPINA, OLGA VIKTOROVNA;SHI, BING;WANG, FANG;WOLCKENHAUER, SCOTT ALAN |
分类号 |
C07D491/052;A61K31/4188;A61P31/14 |
主分类号 |
C07D491/052 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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