发明名称 Heterocyclic janus kinase 3 inhibitors
摘要 The invention relates to compound of the formula (I) or its salt, wherein -R 1 , -R 2 , -R 3 , -R 4 , -R 5 , -M-, -X- and -Y= are as defined in the description, their use of as medicament, the process for their preparation and use for the treatment of JAK3 mediated diseases.
申请公布号 ZA200805605(B) 申请公布日期 2010.02.24
申请号 ZA20080005605 申请日期 2006.12.25
申请人 ASTELLAS PHARMA INC. 发明人 INOUE, TAKAYUKI;TANAKA, AKIRA;NAKAI, KAZUO;SASAKI, HIROSHI;TAKAHASHI, FUMIE;SHIRAKAMI, SHOHEI;HATANAKA, KEIKO;NAKAJIMA, YUTAKA;MUKOYOSHI, KOICHIRO;HAMAGUCHI, HISAO;KUNIKAWA, SHIGEKI;HIGASHI, YASUYUKI
分类号 A61K;A61P;C07D 主分类号 A61K
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