发明名称 CRYSTALLINE SOLVATES OF (1S)-1,5-ANHYDRO-1-C-(3-((PHENYL) METHYL) PHENYL)-D-GLUCITOL DERIVATIVES WITH ALCOHOLS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES
摘要 The present invention relates to physical crystal structures of a compound of the formula I: wherein R 1 , R 2 , R 2a , R 3 and R 4 are as defined herein, especially pharmaceutical compositions containing structures of compound I or II, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures.
申请公布号 EP2069374(A1) 申请公布日期 2009.06.17
申请号 EP20070784499 申请日期 2007.06.21
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 GOUGOUTAS, JACK, Z.;LOBINGER, HILDEGARD;RAMAKRISHNAN, SRIVIDYA;DESHPANDE, PRASHANT, P.;BIEN, JEFFREY, T.;LAI, CHIAJEN;WANG, CHENCHI;RIEBEL, PETER;GROSSO, JOHN, ANTHONY;NIRSCHL, ALEXANDRA, A.;SINGH, JANAK;DIMARCO, JOHN, D.
分类号 C07H7/04;A61K31/70;A61P3/10 主分类号 C07H7/04
代理机构 代理人
主权项
地址