发明名称 PYRAZOLOPYRIMIDINE ANALOGS AND THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS
摘要 The present invention relates to Pyrazolopyrimidine Analogs, methods of making Pyrazolopyrimidine Analogs, compositions comprising a Pyrazolopyrimidine Analog, and methods for treating mTOR-related disorders comprising administering to a subject in need thereof an effective amount of a Pyrazolopyrimidine Analog. The invention also relates to treating PI3K-related disorders comprising administering to a subject in need thereof an effective amount of a Pyrazolopyrimidine Analog.
申请公布号 US2008234262(A1) 申请公布日期 2008.09.25
申请号 US20080050445 申请日期 2008.03.18
申请人 WYETH 发明人 ZASK ARIE;NOWAK PAWEL WOJCIECH;VERHEIJEN JEROEN CUNERA;CURRAN KEVIN J.;KAPLAN JOSHUA;MALWITZ DAVID;BURSAVICH MATTHEW GREGORY;COLE DEREK CECIL;AYRAL-KALOUSTIAN SEMIRAMIS;YU KER;RICHARD DAVID JAMES;LEFEVER MARK
分类号 A61K31/5377;A61K31/519;A61P35/00;C07D413/14;C07D487/04 主分类号 A61K31/5377
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