| 摘要 |
<p>Pharmacol-active heterocyclic cpds. Cpds. of formula shown, where R1 is H, alkyl, alkoxy, NO2, halogen or CF3: R2 is H or alkyl; X is S, SO or SO2; Y is -(CH2)k-N-(CH2)mR3, -(CH2)k-CR4-(CH2)mR5 or -CH=C -(CH2)mR5 where R3 is Ph opt. substd; R4 is H, OH, alkyl, alkoxy, alkanoyl, alkanoyloxy, carbamoyl opt. N- or N,N-alkylated; R5 is H, morpholino, pyrrolidinyl, piperidinyl, hexamethyleneimino, alkyl, cycloalkyl, cycloalkylalkyl, hydroxyalkyl, alkoxyalkyl, Ph or substd. Ph; k is 0 or 1; m is 0-2; n is 3 or 4; are tranquillisers, antipsychotonics, antiemotives, anticonvulsants, antipsychotics, sedatives, analgesics and antihypertensives.</p> |
