发明名称 BIS-PYRIDYLPYRIDONES AS MELANIN-CONCENTRATING HORMONE RECEPTOR 1 ANTAGONISTS
摘要 <p>The invention provides novel bis-pyridylpyridones which are antagonists at the melanin-concentrating hormone receptor 1 (MCHR1 ), pharmaceutical compositions containing them, processes for their preparation, and their use in therapy and for the treatment of obesity and diabetes.</p>
申请公布号 WO2010141539(A1) 申请公布日期 2010.12.09
申请号 WO2010US37010 申请日期 2010.06.02
申请人 GLAXOSMITHKLINE LLC;CHRISTENSEN, SIEGFRIED, BENJAMIN, IV;QIN, DONGHUI;CHEN, SHENGLIN;HUANG, XING;LI, DI;LI, FEI;LI, LEI;LIN, XIAOJUAN;LU, SHI;LU, ZHEN;LV, MAOYUN;WANG, CHUANNING;WU, CHENGDE;XIAO, MEI;YU, HAIYU;ZHANG, WEINA;ZHANG, ZHILIU 发明人 CHRISTENSEN, SIEGFRIED, BENJAMIN, IV;QIN, DONGHUI;CHEN, SHENGLIN;HUANG, XING;LI, DI;LI, FEI;LI, LEI;LIN, XIAOJUAN;LU, SHI;LU, ZHEN;LV, MAOYUN;WANG, CHUANNING;WU, CHENGDE;XIAO, MEI;YU, HAIYU;ZHANG, WEINA;ZHANG, ZHILIU
分类号 A01N43/00;C07D213/06 主分类号 A01N43/00
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